Menene paclitaxel mai ɗaure albumin?

Menene paclitaxel mai ɗaure albumin?Albumin-bound paclitaxel (wanda aka fi sani da albumin paclitaxel, wanda kuma aka rage shi da Nab-P) sabon paclitaxel nanoformulation ne, wanda aka sani da duniya a matsayin mafi haɓakar tsarin paclitaxel.Yana haɗu da albumin ɗan adam endogenous tare da paclitaxel a cikin wani nau'i mara kyau kuma sakamakon nanoparticles gaba ɗaya sun shawo kan rashin lahani na paclitaxel wanda ba zai iya narkewa a cikin ruwa ba, ba tare da buƙatar man fetur na polyoxyethylene castor ko Tween 80 a matsayin haɗin gwiwa ba.Kamar yadda albumin samfurin halitta ne na ƙarshe, yana da fa'idodin kasancewa mai aminci, mara guba, mara lahani, mai yuwuwa, da daidaitawa.

Menene paclitaxel mai ɗaure albumin

Me yasa paclitaxel mai ɗaure albumin shine mafi haɓaka?

1. Babu co-solubilisationno pre-jiyya

Yin amfani da furotin na plasma na asalin halitta, yana ɗaure kwayoyin paclitaxel na hydrophobic a cikin wani nau'i mai ban sha'awa ba tare da wani haɗin gwiwa ba, yana kawar da hypersensitivity da halayen guba wanda ya haifar da haɗin gwiwa, don haka yana kawar da buƙatar pretreatment na hormone kafin amfani da kuma rage lokacin jiko. zuwa mintuna 30, yana rage jinkirin zaman asibiti na majinyatan oncology, har ma da kammala chemotherapy ta asibitin rana.

2. Mafi kyawun magunguna

Idan aka kwatanta da na al'ada paclitaxel, albumin paclitaxel yana da sauri da kuma mafi girma rarraba nama a cikin jiki, kazalika da sannu a hankali excretion daga kyallen takarda, da jurewa kashi a cikin jikin mutum za a iya girma girma da kuma warkewa sakamako da aka muhimmanci inganta.

3. Zabi na gida ƙari tara

Ɗaya daga cikin dalilan da ya sa marasa lafiya da yawa ke jin tsoron cutar sankarau shine cewa rarraba paclitaxel na gargajiya a cikin ƙwayar ƙwayar cuta da sauran kyallen takarda na al'ada daidai ne, yana haifar da sakamako mai tsanani.Sabanin haka, paclitaxel yana da mu'ujiza "zaɓi na haɓaka ƙwayar ƙwayar cuta na gida" kuma maida hankali a cikin ƙwayar ƙwayar cuta ya fi na sauran kyallen takarda na al'ada.

Lura: Abubuwan da za su iya tasiri da aikace-aikacen da aka kwatanta a cikin wannan labarin an ɗauke su daga wallafe-wallafen da aka buga.

Yunnan Hande Bio-Tech Co., Ltd ya kware wajen samar da kayayyakipaclitaxel APIfiye da shekaru 20, kuma yana ɗaya daga cikin manyan masana'antun duniya na paclitaxel API tare da amincewar FDA, takardar shaidar CEP da takardar shaidar GMP a kasar Sin.Hande na iya samar da API mai inganci ba kawai paclitaxel ba har masabis na canja wurin fasaha don paclitaxel albumin.Don ƙarin bayani, da fatan za a tuntuɓe mu a 18187887160.


Lokacin aikawa: Dec-08-2022