Inganci da rawar paclitaxel

Paclitaxel ya fito ne daga Taxus chinensis kuma shine farkon abu da aka samo yana da tasirin hanawa akan ƙwayoyin ƙari.Tsarin paclitaxel yana da wuyar gaske, kuma aikace-aikacensa na likitanci sun fi bayyana a cikin maganin ciwon nono, ciwon huhu, da ciwon daji na ovarian.Paclitaxelwani metabolite ne na biyu da aka fitar daga haushin Taxus chinensis ta masanan kimiya na Amurka, wanda ke da tasiri mai kyau na rigakafin cutar kansa.Bari mu kalli inganci da rawar paclitaxel.

Inganci da rawar paclitaxel

Inganci da rawar dapaclitaxel

1. Anti-tumor sakamako

Paclitaxel magani ne na anti-microtubule antitumor.Paclitaxel na iya inganta taro na microtubule ta hanyar inganta polymerization na spinosomal tubulin subunits, har ma a cikin masu shiga tsakani da ake bukata don taron microtubule na al'ada (kamar GTP, guanosine triphosphate, da dai sauransu)., da dai sauransu) na iya samun wannan tasiri, wanda ya haifar da samuwar microtubules marasa aiki, barga.

2. Maganin ciwon daji

Paclitaxel yana da tasirin anticancer akan layukan ƙwayoyin cuta na sarcoma, cutar sankarar bargo da kuma melanoma.Paclitaxel kuma magani ne na farko ga mata masu fama da ciwon nono da ciwon daji na kwai.Paclitaxel zai iya ɗaure zuwa microtubules, wanda zai iya "daskare" kuma ya hana rabuwa da chromosomes a lokacin rarrabawar kwayar halitta, wanda zai iya kashe kwayoyin cutar kansa da sauri.

3. Maganin ciwon sankarau

Nazarin ya nuna cewa FDA ta amince da paclitaxel don maganin cututtukan cututtuka na rheumatoid, kuma paclitaxel gel wani nau'i ne na kayan aiki na kayan aiki.paclitaxel don maganin cututtuka na rheumatoid.

Lura: Yiwuwar inganci da aikace-aikacen da aka bayyana a cikin wannan labarin an samo su daga wallafe-wallafen da aka buga.

paclitaxel API

Karin karatu:Yunnan Hande Biotechnology Co., Ltd yana mai da hankali kan samar da paclitaxel tsawon shekaru 28.Ita ce masana'anta ta farko mai zaman kanta a duniya na paclitaxel na maganin ciwon daji da aka samo daga shuka wanda FDA ta Amurka, Turai EDQM, TGA ta Australiya, China CFDA, Indiya, Japan da sauran hukumomin kula da ƙasa suka amince.kamfani.Idan kana so ka sayaAPI ɗin Paclitaxel,don Allah a tuntube mu akan layi.


Lokacin aikawa: Satumba-30-2022